Synthesis and anti-Trypanosoma cruzi activity of 3-cyanopyridine derivatives

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ACS Omega - ISSN 2470-1343-9:20 (2024) p. 22360-22370
Auteur(s)
    Brian W. Slafer, Marco A. Dessoy, Ramon G. de Oliveira, Maria C. Mollo, Eun Lee, An Matheeussen, Louis Maes, Guy Caljon, Leonardo L.G. Ferreira, Renata Krogh, Adriano D. Andricopulo, Luiza R. Cruz, Charles E. Mowbray, Jadel M. Kratz, Luiz C. Dias

Synthesis and anti-chagas activity profile of a redox-active lead 3-benzylmenadione revealed by high-content imaging

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ACS Infectious Diseases - ISSN 2373-8227-10:5 (2024) p. 1808-1838
Auteur(s)
    Nathan Trometer, Jeremy Pecourneau, Liwen Feng, Jose A. Navarro-Huerta, Danielle Lazarin-Bidoia, Sueli Oliveira Silva de Lautenschlager, Louis Maes, Amanda Fortes Francisco, John M. Kelly, Brigitte Meunier, Monica Cal, Pascal Maser, Marcel Kaiser, Elisabeth Davioud-Charvet

Chemoselective synthesis and anti-kinetoplastidal properties of 2,6-diaryl-4H-tetrahydro-thiopyran-4-one S-oxides : their interplay in a cascade of redox reactions from diarylideneacetones

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Molecules: a journal of synthetic chemistry and natural product chemistry - ISSN 1420-3049-29:7 (2024) p. 1-25
Auteur(s)
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Lead optimization of the 5-phenylpyrazolopyrimidinone NPD-2975 toward compounds with improved antitrypanosomal efficacy

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Journal of medicinal chemistry - ISSN 0022-2623-67:4 (2024) p. 2849-2863
Auteur(s)
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