Development of biochemical assays to enable FAP-targeted inhibitor discovery and cancer biomarker applications
Source
Antwerp, University of Antwerp, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, Department of Pharmaceutical Sciences, 2026,XVII, 330 p.
In vitro kinetic profiling by enzymatic approaches to select FAPIs with a long residence time
Source
European journal of medicinal chemistry - ISSN 0223-5234-304 (2026) p. 1-19
Selective and orally bioavailable dipeptidyl peptidase 9 inhibitors with potent pyroptosis induction properties
Source
Journal of medicinal chemistry - ISSN 0022-2623-68:21 (2025) p. 23163-23184
Structure-property investigation of new "KetoFAPI" inhibitors of fibroblast activation protein (FAP) : discovery of highly potent, selective compounds with prolonged residence times and promising radiotheranostic potential
Source
Journal of medicinal chemistry - ISSN 0022-2623-68:20 (2025) p. 21739-21765
Synthesis and preclinical evaluation of druglike ¹⁸F-labeled fibroblast activation protein (FAP) inhibitors with enhanced tumor retention
Source
Bioconjugate chemistry - ISSN 1043-1802-36:8 (2025) p. 1887-1906