In vitro kinetic profiling by enzymatic approaches to select FAPIs with a long residence time
Source
European journal of medicinal chemistry - ISSN 0223-5234-304 (2026) p. 1-19
Selective and orally bioavailable dipeptidyl peptidase 9 inhibitors with potent pyroptosis induction properties
Source
Journal of medicinal chemistry - ISSN 0022-2623-68:21 (2025) p. 23163-23184
Using protease inhibitors to prevent intraperitoneal adhesions : effects of nafamostat mesylate, UAMC-00050, GM6001, and enoxaparin in the cecal ligation and puncture model and the ischemic button model
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Surgery today - ISSN 0941-1291- (2025) p.
Structure-property investigation of new "KetoFAPI" inhibitors of fibroblast activation protein (FAP) : discovery of highly potent, selective compounds with prolonged residence times and promising radiotheranostic potential
Source
Journal of medicinal chemistry - ISSN 0022-2623-68:20 (2025) p. 21739-21765
Synthesis and preclinical evaluation of druglike ¹⁸F-labeled fibroblast activation protein (FAP) inhibitors with enhanced tumor retention
Source
Bioconjugate chemistry - ISSN 1043-1802-36:8 (2025) p. 1887-1906