Design, synthesis and stepwise optimization of nitrile-based inhibitors of cathepsins B and L
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Bioorganic and medicinal chemistry - ISSN 0968-0896-29 (2021) p.
Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor
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Bioorganic and medicinal chemistry - ISSN 0968-0896-28:22 (2020) p.
N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S : in silico design, synthesis and biochemical characterization
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Bioorganic and medicinal chemistry letters - ISSN 0960-894X-30:18 (2020) p.
Optimization strategy of single-digit nanomolar cross-class inhibitors of mammalian and protozoa cysteine proteases
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Bioorganic chemistry - ISSN 0045-2068-101 (2020) p.
Mapping the S1 and S1' subsites of cysteine proteases with new dipeptidyl nitrile inhibitors as trypanocidal agents
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PLoS neglected tropical diseases - ISSN 1935-2735-14:3 (2020) p.