Novel quinoline derivatives with broad-spectrum antiprotozoal activities

Source
Archiv der Pharmazie - ISSN 0365-6233- (2024) p.
Author(s)

Synthesis and pharmacological evaluation of fluoro/chloro-substituted acetyl and benzoyl esters of quinine as antimalarial agents

Source
Results in Chemistry - ISSN 2211-7156-7 (2024) p. 1-7
Author(s)
    Jean-Gonfi Mvondo Mbala, Dani Thierry Mawete, Alain Nanikafuako Makiese, Prosper Lwanzo Kwiraviwe, Bibiche Kuyubuka Pangu, Eric Buini Nguimi, Kanyanga Cimanga, Luc Pieters, Gilles Degotte, Michel Frederich, Aristote Matondo, Natascha Van Pelt, Guy Caljon, Bernard Pirotte, Blaise Mbala Mavinga, Sylvie-Mireille Bambi-Nyanguile

DNDI-6174 is a preclinical candidate for visceral leishmaniasis that targets the cytochrome bc₁

Source
Science translational medicine - ISSN 1946-6234-15:726 (2023) p.
Author(s)
    Stéphanie Braillard, Martine Keenan, Karen J. Breese, Jacob Heppell, Michael Abbott, Rafiqul Islam, David M. Shackleford, Kasiram Katneni, Elly Crighton, Gong Chen, Rahul Patil, Given Lee, Karen L. White, Sandra Carvalho, Richard J. Wall, Giulia Chemi, Fabio Zuccotto, Silvia González, Maria Marco, Julianna Deakyne, David Standing, Gino Brunori, Jonathan J. Lyon, Pablo Castañeda-Casado, Isabel Camino, Maria S. Martinez Martinez, Bilal Zulfiqar, Vicky M. Avery, Pim-Bart Feijens, Natascha Van Pelt, An Matheeussen, Sarah Hendrickx, Louis Maes, Guy Caljon, Vanessa Yardley, Susan Wyllie, Susan A. Charman, Eric Chatelain

Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease

Source
European journal of medicinal chemistry - ISSN 0223-5234-246 (2023) p. 1-10
Author(s)
    Celso de Oliveira Rezende, Pablo David Grigol Martinez, Rafael Augusto Alves Ferreira, Paul John Koovits, Bruna Miranda Soares, Leonardo L.G. Ferreira, Simone Michelan-Duarte, Rafael Consolin Chelucci, Adriano D. Andricopulo, An Matheeussen, Natascha Van Pelt, Guy Caljon, Louis Maes, Simon Campbell, Jadel M. Kratz, Charles E. Mowbray, Luiz Carlos Dias