A strategic discovery roadmap towards high-quality leads and drug development candidates for kinetoplastid diseases. Part 2: from molecule to confirmed hit

Source
The journal of antimicrobial chemotherapy - ISSN 0305-7453-81:4 (2026) p. 1-14
Author(s)
    Sarah Hendrickx, Kayhan Ilbeigi, Eli S.J. Thore, Michael G. Bertram, Estefania Calvo-Alvarez, Sener Cintesun, Ana Isabel Olias-Molero, Maria Jesus Corral, Marta Mateo-Barrientos, Jerome Estaquier, Sebastien Pomel, Jose Maria Alunda, Sheraz Gul, Katrien Van Bocxlaer, Frederic Frezard, Joana Tavares, Anabela Cordeiro Da Silva, Maria Paola Costi, Louis Maes, Guy Caljon

Discovery of a series of macrocycles as potent inhibitors of Leishmania infantum

Source
Journal of medicinal chemistry - ISSN 0022-2623-67:20 (2024) p. 18170-18193
Author(s)
    Federico Riu, Larissa Alena Ruppitsch, Duc Duy Vo, Richard S. Hong, Mohit Tyagi, An Matheeussen, Sarah Hendrickx, Vasanthanathan Poongavanam, Guy Caljon, Ahmad Y. Sheikh, Peter Sjo, Jan Kihlberg

In vivo bioluminescence imaging reveals differences in Leishmania infantum parasite killing kinetics by antileishmanial reference drugs

Source
ACS Infectious Diseases - ISSN 2373-8227-10:6 (2024) p. 2101-2107
Author(s)

Q586B2 is a crucial virulence factor during the early stages of Trypanosoma brucei infection that is conserved amongst trypanosomatids

Source
Nature communications - ISSN 2041-1723-15:1 (2024) p. 1-18
Author(s)
    Benoit Stijlemans, Patrick De Baetselier, Inge Van Molle, Laurence Lecordier, Erika Hendrickx, Ema Romão, Cécile Vincke, Wendy Baetens, Steve Schoonooghe, Gholamreza Hassanzadeh-Ghassabeh, Hannelie Korf, Marie Wallays, Joar E. Pinto Torres, David Perez-Morga, Lea Brys, Oscar Campetella, María S. Leguizamón, Mathieu Claes, Sarah Hendrickx, Dorien Mabille, Guy Caljon, Han Remaut, Kim Roelants, Stefan Magez, Jo A. Van Ginderachter, Carl De Trez