Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease

Source
European journal of medicinal chemistry - ISSN 0223-5234-246 (2023) p. 1-10
Author(s)
    Celso de Oliveira Rezende, Pablo David Grigol Martinez, Rafael Augusto Alves Ferreira, Paul John Koovits, Bruna Miranda Soares, Leonardo L.G. Ferreira, Simone Michelan-Duarte, Rafael Consolin Chelucci, Adriano D. Andricopulo, An Matheeussen, Natascha Van Pelt, Guy Caljon, Louis Maes, Simon Campbell, Jadel M. Kratz, Charles E. Mowbray, Luiz Carlos Dias

Supramolecular assembly of pentamidine and polymeric cyclodextrin bimetallic core-shell nanoarchitectures

Source
Beilstein journal of nanotechnology - ISSN 2190-4286-13 (2022) p. 1361-1369
Author(s)
    Alexandru-Milentie Hada, Nina Burduja, Marco Abbate, Claudio Stagno, Guy Caljon, Louis Maes, Nicola Micale, Massimiliano Cordaro, Angela Scala, Antonino Mazzaglia, Anna Pipemo

3-nitroimidazo[1,2-b]pyridazine as a novel scaffold for antiparasitics with sub-nanomolar anti-Giardia lamblia activity

Source
International Journal for Parasitology: Drugs and Drug Resistance - ISSN 2211-3207-19 (2022) p. 47-55
Author(s)
    Yang Zheng, Joachim Müller, Stefan Kunz, Marco Siderius, Louis Maes, Guy Caljon, Norbert Müller, Andrew Hemphill, Geert Jan Sterk, Rob Leurs