Fat or flat? The impact of dipole moment vectors on non-covalent interactions between aromatic tags and macromolecules

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Inorganic Chemistry Frontiers - ISSN 2052-1553- (2025) p.
Auteur(s)
    Josef Holub, Adéla Jílková, Carina Lemke, Lorenzo Cianni, Petra Spiwoková, Martin Horn, Christian Breuer, Adrian Leontovyč, Jiří Brynda, Helena Mertlíková-Kaiserová, Marta Chanová, Fernanda dos Reis Rocho, Carlos A. Montanari, Nelly El-Sakkary, Conor R. Caffrey, Michael Gütschow, Drahomír Hnyk, Michael Mareš, Jindřich Fanfrlík

Novel selective proline-based peptidomimetics for human cathepsin K inhibition

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Bioorganic and medicinal chemistry letters - ISSN 0960-894X-110 (2024) p.
Auteur(s)
    Felipe Cardoso Prado Martins, Fernanda dos Reis Rocho, Vinicius Bonatto, Pedro Henrique Jatai Batista, Jeronimo Lameira, Andrei Leita, Carlos A. Montanari

Differential specificity of SARS-CoV-2 main protease variants on peptide versus protein-based substrates

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The FEBS journal - ISSN 1742-464X-291:1 (2024) p. 61-69
Auteur(s)
    Fernanda dos Reis Rocho, Scott J. Snipas, Anwar Shamim, Wioletta Rut, Marcin Drag, Carlos A. Montanari, Guy S. Salvesen

Nitriles : an attractive approach to the development of covalent inhibitors

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RSC Medicinal Chemistry - ISSN 2632-8682-14:2 (2023) p. 201-217
Auteur(s)
    Vinicius Bonatto, Rafael F. Lameiro, Fernanda dos Reis Rocho, Jeronimo Lameira, Andrei Leitao, Carlos A. Montanari

A patent review on cathepsin K inhibitors to treat osteoporosis (2011-2021)

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Expert opinion on therapeutic patents - ISSN 1354-3776-32:5 (2022) p. 561-573
Auteur(s)
    Fernanda dos Reis Rocho, Vinicius Bonatto, Rafael F. Lameiro, Jeronimo Lameira, Andrei Leitao, Carlos A. Montanari