Immunosuppressive effects of new thiophene-based KV1.3 inhibitors

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European journal of medicinal chemistry - ISSN 0223-5234-259 (2023) p. 1-17
Auteur(s)
    Spela Gubic, Alberto Montalbano, Cesare Sala, Andrea Becchetti, Louise Antonia Hendrickx, Kenny Van Theemsche, Ernesto Lopes Pinheiro-Junior, Ginevra Chioccioli Altadonna, Steve Peigneur, Janez Ilas, Alain J. Labro, Luis A. Pardo, Jan Tytgat, Tihomir Tomasic, Annarosa Arcangeli, Lucija Peterlin Masic

Offsetting voltage-dependent Kv1.5 channel opening through charged residue substitutions on top of the first transmembrane segment

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Bioelectricity - ISSN 2576-3105-4:3 (2022) p. 160-167
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Design of new potent and selective thiophene-based $K_{V}1.3$ inhibitors and their potential for anticancer activity

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Cancers - ISSN 2072-6694-14:11 (2022) p. 1-20
Auteur(s)
    Spela Gubic, Louise Antonia Hendrickx, Xiaoyi Shi, Zan Toplak, Stefan Mozina, Kenny Van Theemsche, Ernesto Lopes Pinheiro-Junior, Steve Peigneur, Alain Labro, Luis A. Pardo, Jan Tytgat, Tihomir Tomasic, Lucija Peterlin Masic

Constitutive, basal, and beta-alanine-mediated activation of the human mas-related G protein-coupled receptor D induces release of the inflammatory cytokine IL-6 and is dependent on NF-kappa B signaling

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International journal of molecular sciences - ISSN 1422-0067-22:24 (2021) p.
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Hydrophobic drug/toxin binding sites in voltage-dependent $K^{+}$and $Na^{+}$channels

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Frontiers in pharmacology - ISSN 1663-9812-11 (2020) p.
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