Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness

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Nature communications - ISSN 2041-1723-10 (2019) p.
Auteur(s)

Comparative genomic analysis of six Glossina genomes, vectors of African trypanosomes

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Genome biology - ISSN 1474-760X-20:1 (2019) p.
Auteur(s)
    Geoffrey M. Attardo, Adly M. Abd-Alla, Alvaro Acosta-Serrano, Guy Caljon, Irina Matetovici, Jan Van Den Abbeele, Adly M. M. Abd-Alla, James E. Allen, Rosemary Bateta, Joshua B. Benoit, Kostas Bourtzis, Jelle Caers, Mikkel B. Christensen, David W. Farrow, Markus Friedrich, Aurelie Hua-Van, Emily C. Jennings, Denis M. Larkin, Daniel Lawson, Michael J. Lehane, Vasileios P. Lenis, Ernesto Lowy-Gallego, Rosaline W. Macharia, Anna R. Malacrida, Heather G. Marco, Daniel Masiga, Gareth L. Maslen, Richard P. Meisel, Irene Meki, Veronika Michalkova, Wolfgang J. Miller, Patrick Minx, Paul O. Mireji, Lino Ometto, Andrew G. Parker, Rita Rio, Clair Rose, Andrew J. Rosendale, Omar Rota-Stabelli, Grazia Savini, Liliane Schoofs, Francesca Scolari, Martin T. Swain, Peter Tak, Chad Tomlinson, George Tsiamis, Aurelien Vigneron, Jingwen Wang, Wesley C. Warren, Serap Aksoy

Revisiting tubercidin against kinetoplastid parasites : aromatic substitutions at position 7 improve activity and reduce toxicity

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European journal of medicinal chemistry - ISSN 0223-5234-164 (2019) p. 689-705
Auteur(s)
    Fabian Hulpia, Gustavo Daniel Campagnaro, Mirko Scortichini, Kristof Van Hecke, Louis Maes, Harry P. de Koning, Guy Caljon, Serge Van Calenbergh

Neutrophils enhance early 'Trypanosoma brucei' infection onset

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Scientific reports - ISSN 2045-2322-8 (2018) p.
Auteur(s)
    Guy Caljon, Dorien Mabille, Benoît Stijlemans, Carl De Trez, Massimiliano Mazzone, Fabienne Tacchini-Cottier, Marie Malissen, Jo A. Van Ginderachter, Stefan Magez, Patrick De Baetselier, Jan Van Den Abeele