5-Aminothiazoles Reveal a New Ligand-Binding Site on Prolyl Oligopeptidase Which is Important for Modulation of Its Protein-Protein Interaction-Derived Functions

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Journal of medicinal chemistry - ISSN 0022-2623
Auteur(s)
    Henri T. Patsi, Tommi P. Kilpelainen, Mikael Jumppanen, Johanna Uhari-Vaananen, Pieter Van Wielendaele, Francesca De Lorenzo, Hengjing Cui, Samuli Auno, Janne Saharinen, Erin Seppala, Nina Sipari, Juha Savinainen, Ingrid De Meester, Anne-Marie Lambeir, Maija Lahtela-Kakkonen, Timo T. Myohanen, Erik A. A. Wallen

Next generation fibroblast activation protein (FAP) targeting PET tracers : the tetrazine ligation allows an easy and convenient way to ¹⁸F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines

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European journal of medicinal chemistry - ISSN 0223-5234-262 (2023) p. 1-10
Auteur(s)