Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity
Botros Sanaa S.   William Samia   Sabra Abdel-Nasser A.   El-Lakkany Naglaa M.   Seif el-Din Sayed H.   García-Rubia Alfonso   Sebastían-Pérez Victor   Blaazer Antoni R.   de Heuvel Erik   Sijm Maarten   Zheng Yang   Garcìa Salado Irene   Munday Jane C.   Maes Louis   de Esch Iwan J.P.   Sterk Geert J.   Augustyns Koen   Leurs Rob   Gil Carmen   De Koning Harry P.  
International Journal for Parasitology: Drugs and Drug Resistance - ISSN 2211-3207-9 (2019) p. 35-43
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DPP8/DPP9 inhibition elicits canonical Nlrp1b inflammasome hallmarks in murine macrophages
Vasconcelos Nathalia M.   Vliegen Gwendolyn   Gonçalves Amanda   De Hert Emilie   Martín-Pérez Rosa   Van Opdenbosch Nina   Jallapally Anvesh   Geiss-Frielander Ruth   Lambeir Anne-Marie   Augustyns Koen   van der Veken Pieter   De Meester Ingrid   Lamkanfi Mohamed  
Life science alliance - ISSN 2575-1077-2:1 (2019)
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α-amino diphenyl phosphonates as novel inhibitors of Escherichia coli ClpP protease
Moreno Cinos Carlos   Sassetti Elisa   Garcìa Salado Irene   Witt Gesa   Benramdane Siham   Reinhardt Laura   Cruz Cristina D.   Joossens Jurgen   van der Veken Pieter   Broetz-Oesterhe Heike   Tammela Paivi   Winterhalter Mathias   Gribbon Philip   Windshuegel Bjoern   Augustyns Koen  
Journal of medicinal chemistry - ISSN 0022-2623-62:2 (2019) p. 774-797
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Synthesis and evaluation of novel benzotropolones as Atg4B inhibiting autophagy blockers
Tanc Muhammet   Cleenewerck Matthias   Kurdi Ammar   Roelandt Ria   Declercq Wim   De Meyer Guido   Augustyns Koen   Martinet Wim   van der Veken Pieter  
Bioorganic chemistry - ISSN 0045-2068-87 (2019) p. 163-168
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ClpP protease, a promising antimicrobial target
Moreno Cinos Carlos   Goossens Kenneth   Garcìa Salado Irene   van der Veken Pieter   De Winter Hans   Augustyns Koen  
International journal of molecular sciences - ISSN 1661-6596-20:9 (2019)
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